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8. 5r and 9. , 9?(Isopropylidenedioxy)?10?benzyloxy?2?benzylsulfanyl?1,2?dehydro? 1?aza?3 Starting with the mixture of the two OZTs 163 and 164 (50mg g, 0.14 mmol) using G.P. 2.3.6. (reaction time 4h), sodium hydrogen carbonate (4.0 eq.) as base and benzyl bromide (4.0 eq.) the compound 166 was obtained after column chromatography on silica gel with a mixture of PE, pp.6-10

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