An efficient route to 5-(hetero)aryl-2,4???- and 2,2???-bipyridines through readily available 3-pyridyl-1,2,4-triazines, Tetrahedron Letters, vol.46, issue.11, p.1791, 2005. ,
DOI : 10.1016/j.tetlet.2005.01.135
Cellule enterocromaffini e cellule basigranulose acidofile nei Vertebrati, Zeitschrift f??r Zellforschung und Mikroskopische Anatomie, vol.1, issue.4, p.743, 1933. ,
DOI : 10.1007/BF02450276
Identification of Enteramine, the Specific Hormone of the Enterochromaffin Cell System, as 5-Hydroxytryptamine, Nature, vol.180, issue.4306, p.800, 1952. ,
DOI : 10.1021/ja01154a551
Crystalline Serotonin, Science, vol.108, issue.2804, p.329, 1948. ,
DOI : 10.1126/science.108.2804.329
8-Hydroxy-2-(dipropylamino)tetralin, a new centrally acting 5-hydroxytryptamine receptor agonist, Journal of Medicinal Chemistry, vol.24, issue.8, p.921, 1981. ,
DOI : 10.1021/jm00140a002
8-Hydroxy-2-(di-n-propylamino)-tetralin discriminates between subtypes of the 5-HT1 recognition site, European Journal of Pharmacology, vol.90, issue.1, p.151, 1983. ,
DOI : 10.1016/0014-2999(83)90230-3
3,4-Dihydro-3-amino-2H-1-benzopyran Derivatives as 5-HT1A Receptor Ligands and Potential Anxiolytic Agents. 1. Synthesis and Structure-Activity Relationship Studies, Journal of Medicinal Chemistry, vol.37, issue.12, p.1779, 1994. ,
DOI : 10.1021/jm00038a007
-1-benzopyran derivatives: synthesis and interaction with serotoninergic receptors, Journal of Pharmacy and Pharmacology, vol.25, issue.7, p.959, 2001. ,
DOI : 10.1211/0022357011776388
URL : https://hal.archives-ouvertes.fr/in2p3-00464800
Substituted 3-amino and/or 3-aminomethyl-3,4-dihydro-2H-1-benzopyrans: synthesis and biological activity, Bioorganic & Medicinal Chemistry, vol.8, issue.3, p.483, 2000. ,
DOI : 10.1016/S0968-0896(99)00311-9
Synthesis of new compounds containing the 2,3-dihydro[1,4]dioxino[2,3-b]pyridine heterocyclic system as a substructure, Tetrahedron, vol.59, issue.20, p.3665, 2003. ,
DOI : 10.1016/S0040-4020(03)00513-1
-1-benzopyran derivatives: synthesis and interaction with serotoninergic receptors, Journal of Pharmacy and Pharmacology, vol.25, issue.7, p.959, 2001. ,
DOI : 10.1211/0022357011776388
URL : https://hal.archives-ouvertes.fr/in2p3-00464800
, and Palladium-Catalyzed N-Heteroarylations, The Journal of Organic Chemistry, vol.69, issue.23, p.7809, 2004. ,
DOI : 10.1021/jo0490898
]pyridines, Journal of Heterocyclic Chemistry, vol.26, issue.5, p.1465, 1986. ,
DOI : 10.1002/jhet.5570230542
Synthesis of functionalized styrenes via palladium-catalyzed coupling of aryl bromides with vinyl tin reagents, The Journal of Organic Chemistry, vol.52, issue.3, p.422, 1987. ,
DOI : 10.1021/jo00379a020
Heck versus suzuki palladium catalysed cross-coupling of a vinylboronate ester with aryl halides., Tetrahedron Letters, vol.34, issue.22, p.3599, 1993. ,
DOI : 10.1016/S0040-4039(00)73646-X
A practical synthesis of the 5-chloromethyl-furo[2,3-b]pyridine pharmacophore, Tetrahedron Letters, vol.36, issue.26, p.4571, 1995. ,
DOI : 10.1016/0040-4039(95)00850-C
Intramolekulare diels-alder-reaktionen mit substituierten 1,2,4,5-tetrazinen und 1,2,4-triazinen, Tetrahedron Letters, vol.26, issue.36, p.4355, 1985. ,
DOI : 10.1016/S0040-4039(00)98733-1
Spiro hydantoin aldose reductase inhibitors derived from 8-aza-4-chromanones, Journal of Medicinal Chemistry, vol.33, issue.7, p.1859, 1990. ,
DOI : 10.1021/jm00169a005
Trifluormethyl-substituierte, heterocyclisch anellierte Pyridine durch intramolekulareDiels-Alder-Cycloaddition mit inversem Elektronenbedarf, Archiv der Pharmazie, vol.321, issue.6, p.349, 1992. ,
DOI : 10.1002/ardp.19923250608
Intramolecular Diels-Alder reactions of 2(1H)-pyrazinones: Synthesis of new Furo/Pyrano-pyridinones and -pyridines, Tetrahedron, vol.51, issue.45, p.12463, 1995. ,
DOI : 10.1016/0040-4020(95)00802-F
Stereochemistry of Electrocyclic Reactions, Journal of the American Chemical Society, vol.87, issue.2, p.395, 1965. ,
DOI : 10.1021/ja01080a054
Diels-Alder reactions of heterocyclic aza dienes. Scope and applications, Chemical Reviews, vol.86, issue.5, p.781, 1986. ,
DOI : 10.1021/cr00075a004
Thermal cycloaddition of dimethyl 1,2,4,5-tetrazine-3,6-dicarboxylate with electron-rich olefins: 1,2-diazine and pyrrole introduction. Preparation of octamethylporphin (OMP), The Journal of Organic Chemistry, vol.49, issue.23, pp.4405-71, 1984. ,
DOI : 10.1021/jo00197a015
Alkaloids Utilizing Sequential Intramolecular Heterocyclic Azadiene Diels???Alder Reactions of an Unsymmetrical 1,2,4,5-Tetrazine, The Journal of Organic Chemistry, vol.65, issue.26, p.9120, 2000. ,
DOI : 10.1021/jo0012546
Intramolekulare Diels-Alder-reaktionen mit 1,2,4-triazinen und 1,2,4,5-tetrazinen zu neuen Siebenring-anellierten pyridinen und pyridazinen., Tetrahedron Letters, vol.27, issue.24, p.2747, 1986. ,
DOI : 10.1016/S0040-4039(00)84633-X
Ketenacetale als dienophile: Reaktivit??t und regiospezifit??t bei (4+2)-cycloadditionen mit inversem elektronenbedarf, Tetrahedron Letters, vol.25, issue.24, p.2541, 1984. ,
DOI : 10.1016/S0040-4039(01)81226-0
4-(??-D-Ribofuranosyl)pyridazine: Neue C-Nukleoside durch [4+2]-Cycloaddition mit inversem Elektronenbedarf, Archiv der Pharmazie, vol.31, issue.6, p.365, 1994. ,
DOI : 10.1002/ardp.19943270604
Cyclization Reactions of 2,2'-Bis-N-methylindolyl to Potential Protein Kinase C Inhibitors, HETEROCYCLES, vol.38, issue.10, p.2267, 1994. ,
DOI : 10.3987/COM-94-6833
Inverse-Electron-Demand Diels-Alder Reactions of Condensed Pyridazines, 5. 1,4-Bis(trifluoromethyl)pyridazino[4,5-b]indole as an Azadiene, HETEROCYCLES, vol.38, issue.8, p.1805, 1994. ,
DOI : 10.3987/COM-94-6726
Intramolecular Diels-Alder reactions of 1,2-diazines: general indoline synthesis. Studies on the preparation of the central and right-hand segments of CC-1065, The Journal of Organic Chemistry, vol.49, issue.12, p.2240, 1984. ,
DOI : 10.1021/jo00186a032
Synthesis of pyridines from dicyanopyrimidines. A diels-alder approach to the c-ring of streptonigrin, Journal of Heterocyclic Chemistry, vol.3, issue.5, p.1111, 1980. ,
DOI : 10.1002/jhet.5570170554
Novel intramolecular Diels-Alder reactions of pyrimidines. Synthesis of heterocyclic annelated pyridines, Tetrahedron Letters, vol.28, issue.14, p.1589, 1987. ,
DOI : 10.1016/S0040-4039(01)81049-2
Synthesis and Reactivity of Some 6-Substituted-2,4-dimethyl-3-pyridinols, a Novel Class of Chain-Breaking Antioxidants, The Journal of Organic Chemistry, vol.69, issue.26, p.9215, 2004. ,
DOI : 10.1021/jo048842u
)-Pyrazinones:?? the Elaboration of a New Tailor-Made Acid-Labile Linker, Journal of Combinatorial Chemistry, vol.5, issue.5, p.560, 2003. ,
DOI : 10.1021/cc0300098
Diels-Alder reaction of heterocyclic azadienes. I. Thermal cycloaddition of 1,2,4-triazine with enamines: simple preparation of substituted pyridines, The Journal of Organic Chemistry, vol.46, issue.10, p.2179, 1981. ,
DOI : 10.1021/jo00323a044
Inverse electron demand Diels-Alder reactions of heterocyclic azadienes. Studies on the total synthesis of lavendamycin: investigative studies on the preparation of the CDE .beta.-carboline ring system and AB quinoline-5,8-quinone ring system, The Journal of Organic Chemistry, vol.50, issue.26, p.5782, 1985. ,
DOI : 10.1021/jo00350a069
Inverse electron demand Diels-Alder reactions of heterocyclic azadienes: formal total synthesis of streptonigrin, Journal of the American Chemical Society, vol.107, issue.20, p.5745, 1985. ,
DOI : 10.1021/ja00306a024
Improved Methodologies for the Preparation of Highly Substituted Pyridines, The Journal of Organic Chemistry, vol.70, issue.24, p.10086, 2005. ,
DOI : 10.1021/jo0518304
Cascade Reactions of Substituted 1,2,4-Triazines:?? Rapid Access to Nitrogen-Containing Polycycles, Journal of the American Chemical Society, vol.126, issue.39, p.12260, 2004. ,
DOI : 10.1021/ja045780g
Indole as a dienophile in inverse electron demand Diels-Alder reactions. 3. Intramolecular reactions with 1,2,4-triazines to access the canthine skeleton, The Journal of Organic Chemistry, vol.57, issue.20, p.5285, 1992. ,
DOI : 10.1021/jo00046a005
A ???one pot??? microwave-mediated synthesis of the basic canthine skeleton: expedient access to unnatural ??-carboline alkaloids, Tetrahedron Letters, vol.44, issue.24, p.4495, 2003. ,
DOI : 10.1016/S0040-4039(03)01019-0
Intramolecular Inverse Electron Demand Diels???Alder Reactions of Tryptamine with Tethered Heteroaromatic Azadienes, Tetrahedron, vol.56, issue.9, p.1165, 2000. ,
DOI : 10.1016/S0040-4020(00)00003-X
Dienophilicity of Imidazole in Inverse Electron Demand Diels-Alder Reactions; Intramolecular Reactions with 1,2,4-Triazines., Tetrahedron Letters, vol.38, issue.43, p.7499, 1997. ,
DOI : 10.1016/S0040-4039(97)01800-5
Intramolecular Inverse-Electron-Demand Diels???Alder Reactions of Imidazoles with 1,2,4-Triazines:?? A New Route to 1,2,3,4-Tetrahydro-1,5-naphthyridines and Related Heterocycles, The Journal of Organic Chemistry, vol.69, issue.21, pp.7171-4345, 2003. ,
DOI : 10.1021/jo040193z
Pyrrole as a dienophile in intramolecular inverse electron-demand Diels-Alder reactions with 1,2,4-triazines, The Journal of Organic Chemistry, vol.58, issue.2, p.516, 1993. ,
DOI : 10.1021/jo00054a044
Cascade reactions of 1,2,4-triazines: direct thermochemical access to functionalized 4,5-dihydroazocines, Tetrahedron Letters, vol.45, issue.47, p.8607, 2004. ,
DOI : 10.1016/j.tetlet.2004.09.169
An efficient route to 5-(hetero)aryl-2,4???- and 2,2???-bipyridines through readily available 3-pyridyl-1,2,4-triazines, Tetrahedron Letters, vol.46, issue.11, p.1791, 2005. ,
DOI : 10.1016/j.tetlet.2005.01.135
Heterodienophilic intramolecular diels-alder reactions of 1,2,4 triazines., Tetrahedron, vol.43, issue.21, p.5159, 1987. ,
DOI : 10.1016/S0040-4020(01)87691-2
Intramolecular Diels-Alder reactions of 1,2,4-triazines. Routes to condensed pyrazines via cycloaddition of nitrile dienophiles, The Journal of Organic Chemistry, vol.54, issue.6, p.1245, 1989. ,
DOI : 10.1021/jo00267a006
1,2,4-triazines in organic synthesis. 8. Intramolecular diels-alder reaction of 5-acyl-1,2,4-triazineoxime ethers. New route of synthesis of alkylhetarylketones, Chemistry of Heterocyclic Compounds, vol.97, issue.3, p.334, 1999. ,
DOI : 10.1007/BF02259365
A new and simple ???LEGO??? system for the synthesis of branched oligopyridines, Tetrahedron Letters, vol.39, issue.37, p.6691, 1998. ,
DOI : 10.1016/S0040-4039(98)01438-5
A new and simple ???LEGO??? system for the synthesis of 2,6-oligopyridines, Tetrahedron Letters, vol.39, issue.37, p.6687, 1998. ,
DOI : 10.1016/S0040-4039(98)01437-3
The preparation of 1,2,4-triazines from ??,??-diketo-ester equivalents and their application in pyridine synthesis, Tetrahedron Letters, vol.46, issue.36, p.6111, 2005. ,
DOI : 10.1016/j.tetlet.2005.06.163
Intramolecular Diels-Alder reactions of 1,2,4-triazines. A facile synthesis of thieno[2,3-b]pyridines and 3,4-dihydro-2H-thiopyrano[2,3-b]pyridines, The Journal of Organic Chemistry, vol.52, issue.19, p.4280, 1987. ,
DOI : 10.1021/jo00228a023
Diels-Alder reactions of 1,2,4-triazines. Synthesis of thieno[2,3-c]pyridines and 3,4-dihydro-2H-thiopyrano[2,3-c]pyridines from 6-(alkynylthio)-1,2,4-triazines, The Journal of Organic Chemistry, vol.54, issue.21, p.4984, 1989. ,
DOI : 10.1021/jo00282a006
Novel cycloaddition routes to fused heterocycles, Bulletin des Soci??t??s Chimiques Belges, vol.97, issue.8-9, p.599, 1988. ,
DOI : 10.1002/bscb.19880970803
Further intramolecular diels-alder reactions of 1,2,4-triazines. Synthesis of dihydropyrrolo[2,3-]pyridines, Tetrahedron Letters, vol.28, issue.4, p.379, 1987. ,
DOI : 10.1016/S0040-4039(00)95733-2
Intramolecular Diels-Alder reactions of 1,2,4-triazines. Synthesis of condensed pyrimidines, The Journal of Organic Chemistry, vol.52, issue.19, p.4287, 1987. ,
DOI : 10.1021/jo00228a024
Tandem Vicarious Nucleophilic Substitution of Hydrogen/Intramolecular Diels???Alder Reaction of 1,2,4-Triazines into Functionalized Cycloalkenopyridines, CHEMICAL & PHARMACEUTICAL BULLETIN, vol.50, issue.4, p.463, 2002. ,
DOI : 10.1248/cpb.50.463
Intramolecular Diels-Alder reactions of 1,2,4-triazines. Synthesis of 2,3-cyclopentenopyridines and 5,6,7,8-tetrahydroquinolines, The Journal of Organic Chemistry, vol.56, issue.5, p.1807, 1991. ,
DOI : 10.1021/jo00005a027
Synthesis of isoquinolines by cycloaddition of arynes to 1,2,4-triazines, Tetrahedron, vol.48, issue.33, p.6821, 1992. ,
DOI : 10.1016/S0040-4020(01)89873-2
1,2,4-triazines. III. A convenient synthesis of 1,2,4-triazines and their covalent hydration, Journal of Heterocyclic Chemistry, vol.1, issue.4, p.767, 1970. ,
DOI : 10.1002/jhet.5570070403
-1,2,4-triazole (guanazine) and its 4-arylideneamino derivatives, Journal of Heterocyclic Chemistry, vol.58, issue.II, p.1077, 1989. ,
DOI : 10.1002/jhet.5570260431
URL : https://hal.archives-ouvertes.fr/hal-00283069
Trimerization of Imidates, The Journal of Organic Chemistry, vol.26, issue.8, p.2778, 1961. ,
DOI : 10.1021/jo01066a036
Intramolecular diels-alder reactions of 1,2,4-triazines., Tetrahedron, vol.43, issue.21, p.5145, 1987. ,
DOI : 10.1016/S0040-4020(01)87690-0
An Efficient Intermolecular Palladium-Catalyzed Synthesis of Aryl Ethers, Journal of the American Chemical Society, vol.123, issue.43, p.10770, 2001. ,
DOI : 10.1021/ja016863p
Palladium Alkoxides:?? Potential Intermediacy in Catalytic Amination, Reductive Elimination of Ethers, and Catalytic Etheration. Comments on Alcohol Elimination from Ir(III), Journal of the American Chemical Society, vol.118, issue.51, p.13109, 1996. ,
DOI : 10.1021/ja963273w
-Isoprostanes, Journal of the American Chemical Society, vol.124, issue.44, p.13121, 2002. ,
DOI : 10.1021/ja020816v
URL : https://hal.archives-ouvertes.fr/hal-01447465
Total Synthesis of Apoptolidin:?? Construction of Enantiomerically Pure Fragments, Journal of the American Chemical Society, vol.125, issue.50, p.15433, 2003. ,
DOI : 10.1021/ja0304953
-Protection of the Uracil Base and Hybridization Properties of Oligonucleotides Incorporating These Modified Nucleoside Derivatives, The Journal of Organic Chemistry, vol.68, issue.26, p.9971, 2003. ,
DOI : 10.1021/jo035246b
Diastereoselective Synthesis of Substituted Tetrahydroquinoline-4-carboxylic Esters by a Tandem Reduction???Reductive Amination Reaction, The Journal of Organic Chemistry, vol.66, issue.8, p.2822, 2001. ,
DOI : 10.1021/jo001761n
Intramolecular Diels-Alder reactions of 1,2,4-triazines. Routes to condensed pyrazines via cycloaddition of nitrile dienophiles, The Journal of Organic Chemistry, vol.54, issue.6, p.1245, 1989. ,
DOI : 10.1021/jo00267a006
Novel intramolecular diels-alder reactions with alkynylthio derivatives of 1,2,4-triazines. New routes to thieno[2,3-]pyridines and thieno[2,3-]pyridines., Tetrahedron Letters, vol.26, issue.20, p.2419, 1985. ,
DOI : 10.1016/S0040-4039(00)94842-1
Synthesis of 7-azaindole and 7-azaoxindole derivatives through a palladium-catalyzed cross-coupling reaction, The Journal of Organic Chemistry, vol.57, issue.25, p.6995, 1992. ,
DOI : 10.1021/jo00051a062
Stereocontrolled Synthesis of the Diene and Triene Macrolactones of Oximidines I and II:??? Organometallic Coupling versus Standard Macrolactonization, Organic Letters, vol.3, issue.22, p.3487, 2001. ,
DOI : 10.1021/ol016744e
An efficient method for synthesis of ??-keto acid esters from terminal alkynes, Tetrahedron Letters, vol.43, issue.13, p.2427, 2002. ,
DOI : 10.1016/S0040-4039(02)00290-3
Novel and convenient method for the stereo- and regiospecific synthesis of conjugated alkadienes and alkenynes via the palladium-catalyzed cross-coupling reaction of 1-alkenylboranes with bromoalkenes and bromoalkynes, Journal of the American Chemical Society, vol.107, issue.4, p.972, 1985. ,
DOI : 10.1021/ja00290a037
Prim, Les complexes de palladium en synthèse organique, CNRS Editions, 2001. ,
Palladium-Catalyzed Chemoselective Cross-Coupling of Acyl Chlorides and Organostannanes, The Journal of Organic Chemistry, vol.70, issue.21, p.8601, 2005. ,
DOI : 10.1021/jo051257o
Large rate accelerations in the stille reaction with tri-2-furylphosphine and triphenylarsine as palladium ligands: mechanistic and synthetic implications, Journal of the American Chemical Society, vol.113, issue.25, p.9585, 1991. ,
DOI : 10.1021/ja00025a025
On the Nature of the "Copper Effect" in the Stille Cross-Coupling, The Journal of Organic Chemistry, vol.59, issue.20, p.5905, 1994. ,
DOI : 10.1021/jo00099a018
Quantitative Evaluation of the Factors Contributing to the ???Copper Effect??? in the Stille Reaction, Organometallics, vol.22, issue.6, p.1305, 2003. ,
DOI : 10.1021/om020896b
Efficient and practical method for synthesizing optically active ??-trityloxymethyl-??-alkylidene-??-butyrolactones using Ti(II)-mediated intramolecular nucleophilic acyl substitution reaction, Tetrahedron Letters, vol.39, issue.43, p.7947, 1998. ,
DOI : 10.1016/S0040-4039(98)01769-9
An efficient method for the alkynylation of oxiranes using alkynyl boranes, Tetrahedron Letters, vol.24, issue.4, p.391, 1983. ,
DOI : 10.1016/S0040-4039(00)81416-1
Selective Synthesis of Functionalized, Tertiary Silanes by Diastereoselective Rearrangement???Addition, Organic Letters, vol.7, issue.22, p.4911, 2005. ,
DOI : 10.1021/ol0518636
]thienyloxy)-2-propanols, Journal of Heterocyclic Chemistry, vol.70, issue.5, p.937, 1980. ,
DOI : 10.1002/jhet.5570170518
Efficient synthesis of 2- and 3-substituted-2,3-dihydro [1,4]dioxino[2,3-b]pyridine derivatives, Tetrahedron, vol.60, issue.31, p.6461, 2004. ,
DOI : 10.1016/j.tet.2004.06.041
Boron trifluoride assisted opening of epoxides by lithium alkenyl aluminate reagents, Tetrahedron, vol.45, issue.19, p.6197, 1989. ,
DOI : 10.1016/S0040-4020(01)85130-9